Org 27569 kinase inhibitor product blog
Tags: Kinase Inhibitor; Org 27569; Org 27569 kinase inhibitor;
The Org 27569 n/a (Catalog #MBS8506234) is an Inhibitor and is intended for research purposes only. The product is available for immediate purchase.To buy or view more detailed product information and pricing, please click on the technical datasheet page below:
Please refer to the product datasheet for known applications of a given inhibitor. We\'ve tested the Org 27569 with the following immunoassay(s):
Testing Data
Org 27569 is an allosteric modulator of CB1 cannabinoid receptor. It significantly increases the binding of CB1 receptor agonist [3H]-CP 55, 940 (pKB = 5.67) and causes a significant decrease in specific binding of CB1 receptor inverse agonist SR141716A (Rimonabant; pKB = 5.95); in the reporter gene assay behaves as insurmountable CP 55, 940 antagonist; pKB = 7.57 at CB1 receptors in mouse vas deferens. [1][2].
Formula: C24H28ClN3O
CAS Number: 868273-06-7.