GSK343 inhibitor product blog
Tags: Inhibitor; GSK343; GSK343 inhibitor;
The GSK343 n/a (Catalog #MBS578634) is an Inhibitor and is intended for research purposes only. The product is available for immediate purchase.To buy or view more detailed product information and pricing, please click on the technical datasheet page below:
Please refer to the product datasheet for known applications of a given inhibitor. We\'ve tested the GSK343 with the following immunoassay(s):
Structure
GSK343 is a potent and selective EZH2 inhibitor with IC50 of 4 nM, showing 60 fold selectivity against EZH1, and >1000 fold selectivity against other histone methyltransferases.
CAS: 1346704-33-3
Smiles: CCCc1c(c(=O)[nH]c(c1)C)CNC(=O)c1c2cnn(c2cc(c1)c1cc(ncc1)N1CCN(CC1)C)C(C)C. Formula: C31H39N7O2.