Exp3174 inhibitor product blog
Tags: Inhibitor; Exp3174; Exp3174 inhibitor;
The Exp3174 n/a (Catalog #MBS579591) is an Inhibitor and is intended for research purposes only. The product is available for immediate purchase.To buy or view more detailed product information and pricing, please click on the technical datasheet page below:
Please refer to the product datasheet for known applications of a given inhibitor. We\'ve tested the Exp3174 with the following immunoassay(s):
Structure
CAS: 124750-92-1
Formula: C22H21ClN6O2
Pathways: Endocrinology/Hormones
Smiles: c1(n(c(c(n1)Cl)C(=O)O)Cc1ccc(cc1)c1c(cccc1)c1n[nH]nn1)CCCC. Receptor: AT1 receptor
Bioactivity: EXP-3174 is a potent AT1 antagonist (Kis = 0.57 and 0.67 nM for rat and human forms, respectively), producing a depressor response and vasodilatation.
Solubility: DMSO: Soluble
Solubility Note: For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.